| Constraining cyclic peptides to mimic protein structure motifs TA Hill, NE Shepherd, F Diness, DP Fairlie Angewandte Chemie International Edition 53 (48), 13020-13041, 2014 | 481 | 2014 |
| Systemic delivery of peptides by the oral route: Formulation and medicinal chemistry approaches DJ Brayden, TA Hill, DP Fairlie, S Maher, RJ Mrsny Advanced drug delivery reviews 157, 2-36, 2020 | 253 | 2020 |
| A novel class of anticancer compounds targets the actin cytoskeleton in tumor cells JR Stehn, NK Haass, T Bonello, M Desouza, G Kottyan, H Treutlein, ... Cancer research 73 (16), 5169-5182, 2013 | 220 | 2013 |
| Comparative α‐Helicity of cyclic pentapeptides in water AD De Araujo, HN Hoang, WM Kok, F Diness, P Gupta, TA Hill, RW Driver, ... Angewandte Chemie International Edition 53 (27), 6965-6969, 2014 | 210 | 2014 |
| Downsizing human, bacterial, and viral proteins to short water-stable alpha helices that maintain biological potency RS Harrison, NE Shepherd, HN Hoang, G Ruiz-Gómez, TA Hill, ... Proceedings of the National Academy of Sciences 107 (26), 11686-11691, 2010 | 208 | 2010 |
| Inhibition of Dynamin Mediated Endocytosis by the DynolesSynthesis and Functional Activity of a Family of Indoles TA Hill, CP Gordon, AB McGeachie, B Venn-Brown, LR Odell, N Chau, ... Journal of medicinal chemistry 52 (12), 3762-3773, 2009 | 195 | 2009 |
| Improving on nature: making a cyclic heptapeptide orally bioavailable DS Nielsen, HN Hoang, RJ Lohman, TA Hill, AJ Lucke, DJ Craik, ... Angewandte Chemie International Edition 53 (45), 12059-12063, 2014 | 168 | 2014 |
| Heterocyclic substituted cantharidin and norcantharidin analogues—synthesis, protein phosphatase (1 and 2A) inhibition, and anti-cancer activity TA Hill, SG Stewart, B Sauer, J Gilbert, SP Ackland, JA Sakoff, ... Bioorganic & medicinal chemistry letters 17 (12), 3392-3397, 2007 | 129 | 2007 |
| Norcantharimides, synthesis and anticancer activity: Synthesis of new norcantharidin analogues and their anticancer evaluation TA Hill, SG Stewart, SP Ackland, J Gilbert, B Sauer, JA Sakoff, ... Bioorganic & medicinal chemistry 15 (18), 6126-6134, 2007 | 125 | 2007 |
| Green chemistry approaches to the Knoevenagel condensation: comparison of ethanol, water and solvent free (dry grind) approaches A McCluskey, PJ Robinson, T Hill, JL Scott, JK Edwards Tetrahedron letters 43 (17), 3117-3120, 2002 | 112 | 2002 |
| Crystal structures of protein-bound cyclic peptides AK Malde, TA Hill, A Iyer, DP Fairlie Chemical Reviews 119 (17), 9861-9914, 2019 | 107 | 2019 |
| Update 1 of: Beta-Strand Mimetics Wendy A. Loughlin, Joel D. A. Tyndall, Matthew P. Glenn,Timothy A. Hill ... Chemical Reviews 110 (6), PR32-PR69, 2010 | 104* | 2010 |
| Small molecule inhibitors of dynamin I GTPase activity: development of dimeric tyrphostins T Hill, LR Odell, JK Edwards, ME Graham, AB McGeachie, J Rusak, ... Journal of medicinal chemistry 48 (24), 7781-7788, 2005 | 92 | 2005 |
| Flexibility versus rigidity for orally bioavailable cyclic hexapeptides DS Nielsen, RJ Lohman, HN Hoang, TA Hill, A Jones, AJ Lucke, ... ChemBioChem 16 (16), 2289-2293, 2015 | 76 | 2015 |
| Norcantharidin analogues: synthesis, anticancer activity and protein phosphatase 1 and 2A inhibition TA Hill, SG Stewart, CP Gordon, SP Ackland, J Gilbert, B Sauer, JA Sakoff, ... ChemMedChem: Chemistry Enabling Drug Discovery 3 (12), 1878-1892, 2008 | 76 | 2008 |
| Cyclic Penta- and Hexaleucine Peptides without N-Methylation Are Orally Absorbed TA Hill, RJ Lohman, HN Hoang, DS Nielsen, CCG Scully, WM Kok, L Liu, ... ACS medicinal chemistry letters 5 (10), 1148-1151, 2014 | 73 | 2014 |
| Long chain amines and long chain ammonium salts as novel inhibitors of dynamin GTPase activity TA Hill, LR Odell, A Quan, R Abagyan, G Ferguson, PJ Robinson, ... Bioorganic & Medicinal Chemistry Letters 14 (12), 3275-3278, 2004 | 72 | 2004 |
| Iminochromene inhibitors of dynamins I and II GTPase activity and endocytosis TA Hill, A Mariana, CP Gordon, LR Odell, MJ Robertson, AB McGeachie, ... Journal of medicinal chemistry 53 (10), 4094-4102, 2010 | 70 | 2010 |
| Connecting hydrophobic surfaces in cyclic peptides increases membrane permeability HN Hoang, TA Hill, DP Fairlie Angewandte Chemie 133 (15), 8466-8471, 2021 | 63 | 2021 |
| Truncated and helix-constrained peptides with high affinity and specificity for the cFos coiled-coil of AP-1 T Rao, G Ruiz-Gomez, TA Hill, HN Hoang, DP Fairlie, JM Mason PLoS One 8 (3), e59415, 2013 | 61 | 2013 |
David P FairlieProfessor, University of Queensland, Brisbane, AustraliaVerified email at imb.uq.edu.au
