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FI935867A0 - Tetrahydrobensazepinderivat som inhibiterar lipoxigenas - Google Patents

Tetrahydrobensazepinderivat som inhibiterar lipoxigenas

Info

Publication number
FI935867A0
FI935867A0 FI935867A FI935867A FI935867A0 FI 935867 A0 FI935867 A0 FI 935867A0 FI 935867 A FI935867 A FI 935867A FI 935867 A FI935867 A FI 935867A FI 935867 A0 FI935867 A0 FI 935867A0
Authority
FI
Finland
Prior art keywords
alkyl
pct
sec
lipoxygenase
arylalkyl
Prior art date
Application number
FI935867A
Other languages
English (en)
Finnish (fi)
Other versions
FI935867L (fi
FI935867A7 (fi
Inventor
Takafumi Ikeda
Yoko Hoshino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI935867L publication Critical patent/FI935867L/fi
Publication of FI935867A0 publication Critical patent/FI935867A0/fi
Publication of FI935867A7 publication Critical patent/FI935867A7/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D223/00Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16Benzazepines; Hydrogenated benzazepines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Hydrogenated Pyridines (AREA)
FI935867A 1991-06-28 1992-05-27 Tetrahydrobentsatsepiini-johdannaisia, jotka estävät lipoksygenaasia FI935867A7 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP3158832A JPH0717612B2 (ja) 1991-06-28 1991-06-28 新規なテトラヒドロベンズアゼピン誘導体
PCT/US1992/004197 WO1993000335A1 (fr) 1991-06-28 1992-05-27 Derives de la tetrahydrobenzazepine inhibant la lipoxygenase

Publications (3)

Publication Number Publication Date
FI935867L FI935867L (fi) 1993-12-27
FI935867A0 true FI935867A0 (fi) 1993-12-27
FI935867A7 FI935867A7 (fi) 1993-12-27

Family

ID=15680372

Family Applications (1)

Application Number Title Priority Date Filing Date
FI935867A FI935867A7 (fi) 1991-06-28 1992-05-27 Tetrahydrobentsatsepiini-johdannaisia, jotka estävät lipoksygenaasia

Country Status (13)

Country Link
US (1) US5478822A (fr)
EP (1) EP0591255B1 (fr)
JP (1) JPH0717612B2 (fr)
AT (1) ATE132857T1 (fr)
CA (1) CA2111460C (fr)
DE (1) DE69207597T2 (fr)
DK (1) DK0591255T3 (fr)
ES (1) ES2082474T3 (fr)
FI (1) FI935867A7 (fr)
GR (1) GR3019196T3 (fr)
IE (1) IE70234B1 (fr)
PT (1) PT100628A (fr)
WO (1) WO1993000335A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2167715C (fr) * 1993-07-20 1998-10-06 Akiyoshi Kawai Hydroxyurees heteroaryliques cycloalcenyliques
WO1998006701A1 (fr) * 1996-08-15 1998-02-19 Smithkline Beecham Corporation Antagonistes du recepteur de l'il-8
EP1056187A4 (fr) 1998-02-13 2005-11-02 Yaskawa Denki Seisakusho Kk Moteur lineaire
US7229986B2 (en) 2000-05-16 2007-06-12 Takeda Pharmaceutical Company Ltd. Melanin-concentrating hormone antagonist

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ215487A (en) * 1985-03-16 1990-01-29 Wellcome Found Aryl derivatives, pharmaceutical compositions thereof and preservation of cut flowers
EP0279263B1 (fr) * 1987-02-10 1993-08-04 Abbott Laboratories Composés inhibant la lipoxygénase, contenant de l'indole, du benzofurane ou du benzothiophène
ES2053609T3 (es) * 1987-04-24 1994-08-01 Abbott Lab Derivados de urea inhibidores de lipoxigenasa.
US4981865A (en) * 1989-05-26 1991-01-01 Warner-Lambert Co. N-hydroxyamide, N-hydroxythioamide, hydroxyurea, and N-hydroxythiourea derivatives of selected nsaids as antiinflammatory agents

Also Published As

Publication number Publication date
EP0591255B1 (fr) 1996-01-10
EP0591255A1 (fr) 1994-04-13
IE922075A1 (en) 1992-12-30
US5478822A (en) 1995-12-26
DE69207597T2 (de) 1996-05-23
CA2111460A1 (fr) 1993-01-07
FI935867L (fi) 1993-12-27
WO1993000335A1 (fr) 1993-01-07
JPH059181A (ja) 1993-01-19
ATE132857T1 (de) 1996-01-15
PT100628A (pt) 1993-09-30
ES2082474T3 (es) 1996-03-16
GR3019196T3 (en) 1996-06-30
IE70234B1 (en) 1996-11-13
DK0591255T3 (da) 1996-02-12
FI935867A7 (fi) 1993-12-27
DE69207597D1 (de) 1996-02-22
CA2111460C (fr) 1996-11-19
JPH0717612B2 (ja) 1995-03-01

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